oral-dog LD50 500 mg/kg "Psychotropic Drugs and Related Compounds," 2nd ed., Usdin, E., and D.H. Efron, Washington, DC, 1972Vol. -, Pg. 436, 1972.
oral-human TDLo 4111 mg/kg GASTROINTESTINAL: OTHER CHANGES
BEHAVIORAL: TREMOR
BEHAVIORAL: MUSCLE WEAKNESS New England Journal of Medicine. Vol. 287, Pg. 867, 1972.
oral-man TDLo 8 mg/kg GASTROINTESTINAL: NAUSEA OR VOMITING
SKIN AND APPENDAGES (SKIN): "DERMATITIS, OTHER: AFTER SYSTEMIC EXPOSURE" American Journal of Psychiatry. Vol. 141, Pg. 909, 1984.
oral-man TDLo 54 mg/kg BEHAVIORAL: SLEEP
BEHAVIORAL: "HALLUCINATIONS, DISTORTED PERCEPTIONS" New Zealand Medical Journal. Vol. 97, Pg. 23, 1984.
oral-man TDLo 1080 mg/kg/13W SKIN AND APPENDAGES (SKIN): "DERMATITIS, ALLERGIC: AFTER SYSTEMIC EXPOSURE" Journal of Clinical Psychiatry. Vol. 47, Pg. 330, 1986.
oral-man TDLo 25000 mg/kg/4Y-I BEHAVIORAL: TREMOR
SENSE ORGANS AND SPECIAL SENSES: MIOSIS (PUPILLARY CONSTRICTION): EYE Journal of Clinical Psychiatry. Vol. 46, Pg. 292, 1985.
intraperitoneal-mouse LD50 236 mg/kg BEHAVIORAL: ATAXIA
BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX)
BEHAVIORAL: EXCITEMENT Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
intravenous-mouse LD50 497 mg/kg LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION
BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX) Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
oral-mouse LD50 531 mg/kg Russian Pharmacology and Toxicology Vol. 33, Pg. 266, 1970.
intraperitoneal-rat LD50 156 mg/kg GASTROINTESTINAL: "HYPERMOTILITY, DIARRHEA"
LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION
BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
intravenous-rat LD50 241 mg/kg BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX)
LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
oral-rat LD50 525 mg/kg LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION
BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY)
GASTROINTESTINAL: "HYPERMOTILITY, DIARRHEA" Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
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subcutaneous-mouse LD50 413 mg/kg Russian Pharmacology and Toxicology Vol. 33, Pg. 266, 1970.
subcutaneous-rat LD50 434 mg/kg SENSE ORGANS AND SPECIAL SENSES: LACRIMATION: EYE
LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION
SKIN AND APPENDAGES (SKIN): HAIR: OTHER Kiso to Rinsho. Clinical Report. Vol. 7, Pg. 1273, 1973.
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